For licensed healthcare professionals. The protocol figures below are drawn from published labeling and peer-reviewed literature for educational reference. They are not a prescription, not a recommendation, and not a substitute for the dispensing pharmacy's labeling or your own clinical judgment.
Sexual Health

PT-141

aka Bremelanotide, Vyleesi
FDA approved Not WADA-listed

Melanocortin receptor agonist FDA-approved for hypoactive sexual desire disorder in premenopausal women. SC injection on-demand.

At a glance

Common vial size
10 mg
Reference dose
1.75 mg
Frequency
PRN — max 1 dose/24 h, 8 doses/month

Reference titration protocol

500 mcg × 8 wks → 1000 mcg × 4 wks → 1500 mcg × 4 wks, once daily.

Reference titration ladder for PT-141
StepDoseDurationAdministrations / week
1500 mcg4 weeks7×
21 mg4 weeks7×
31.5 mg4 weeks7×
Reconstitution example

A 10 mg vial reconstituted with 3 mL of bacteriostatic water yields 3.333 mg/mL. Confirm the diluent and volume against the labeling that ships with the vial.

Open this configuration in the calculator

Clinical notes

  • Transient BP elevation — avoid in uncontrolled hypertension

Available formulations

Presentations carried across the VitaRelay pharmacy network, including 503A compounded, 503B outsourcing facility, and research & development sourcing. Pricing and state-level availability are shown to verified accounts only.

  • Injectable503A
  • Lyophilized PowderR&D
  • Nasal Spray503A
  • Pen503B

References

Pricing and ordering are for verified accounts

VitaRelay serves licensed practices, prescribers, and pharmacies. Catalog pricing, availability by state, and ordering are available after your account is verified.

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