For licensed healthcare professionals. The protocol figures below are drawn from published labeling and peer-reviewed literature for educational reference. They are not a prescription, not a recommendation, and not a substitute for the dispensing pharmacy's labeling or your own clinical judgment.

Metabolic

Tesofensine

Investigational Not WADA-listed

Triple monoamine reuptake inhibitor in Phase III for obesity (TIPO-4). Oral, once daily.

At a glance

Common vial size: Not vial-based
Reference dose: 500 mcg
Frequency: Once daily, oral

Reference titration protocol

Oral 0.25 mg QD × 4 wks → 0.5 mg → 1.0 mg; monitor HR/BP at higher doses.

Reference titration ladder for Tesofensine
Step	Dose	Duration	Administrations / week
1	250 mcg	4 weeks	7×
2	500 mcg	4 weeks	7×
3	750 mcg	4 weeks	7×
4	1 mg	4 weeks	7×

Available formulations

Presentations carried across the VitaRelay pharmacy network, including 503A compounded, 503B outsourcing facility, and research & development sourcing. Pricing and state-level availability are shown to verified accounts only.

Capsule/TabletR&D
Capsule/Tablet503A
Capsules503A

References

Astrup et al., Lancet 2008

Pricing and ordering are for verified accounts

VitaRelay serves licensed practices, prescribers, and pharmacies. Catalog pricing, availability by state, and ordering are available after your account is verified.

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AICAR

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Mitochondrial-derived peptide implicated in metabolic homeostasis and insulin sensitivity. Preclinical/early human research only.

Educational information for licensed healthcare professionals

The material on this page is general educational information intended for licensed healthcare professionals and their clinical staff. It is not medical advice, is not a substitute for professional judgment, and does not establish a provider-patient relationship. Nothing here should be read as a recommendation for, or endorsement of, any specific therapy, product, or course of treatment. Compounded preparations must be handled in accordance with applicable federal and state law, the dispensing pharmacy's labeling, and your own institutional policies. All clinical decisions — including product selection, preparation, dosing, and administration — remain the sole responsibility of the treating licensed practitioner.

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